TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:TP_TRANSPORTER: inhibition of ochratoxin A uptake (ochratoxin A / 1uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Rattus norvegicus)
Kyoto University Hospital
Curated by ChEMBL
Kyoto University Hospital
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:TP_TRANSPORTER: inhibition of MTX uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 850nMAssay Description:TP_TRANSPORTER: inhibition of Adefovir uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of Adefovir uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:TP_TRANSPORTER: inhibition of 6-Carboxyfluorescein uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:TP_TRANSPORTER: inhibition of Adefovir uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of Adefovir uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human OAT1More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of OAT1 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of Adefovir uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of OAT1 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 4.60E+3nMAssay Description:TP_TRANSPORTER: inhibition of Urate uptake (Urate: 300 uM) in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 4.90E+3nMAssay Description:TP_TRANSPORTER: inhibition of 6-Carboxyfluorescein uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:TP_TRANSPORTER: inhibition of Adefovir uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of Adefovir uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 6.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of 6-Carboxyfluorescein uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 7.40E+3nMAssay Description:TP_TRANSPORTER: inhibition of Adefovir uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of Adefovir uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of OAT1 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 8.80E+3nMAssay Description:TP_TRANSPORTER: inhibition of 6-Carboxyfluorescein uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 9.90E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 9.90E+3nMAssay Description:TP_TRANSPORTER: trans-stimulation in OAT1-COS7 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.21E+4nMAssay Description:Inhibition of OAT1 (unknown origin)More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.23E+4nMAssay Description:TP_TRANSPORTER: inhibition of PHA uptake (PHA: 5uM) in hOAT1-expressing S2 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.25E+4nMAssay Description:TP_TRANSPORTER: inhibition of Urate uptake (Urate: 300 uM) in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of human OAT1 expressed in HEK293 cells assessed as P-amino hippuric acid uptake inhibition incubated for 10 mins by UPLC-MS/MS methodMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.83E+4nMAssay Description:Inhibition of OAT1 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in OAT-expressing OK cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 2.05E+4nMAssay Description:TP_TRANSPORTER: inhibition of Adefovir uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 2.33E+4nMAssay Description:Inhibition of OAT1 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in OAT1-expressing OK cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 2.70E+4nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in OAT-expressing OK cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 2.80E+4nMAssay Description:TP_TRANSPORTER: inhibition of 6-Carboxyfluorescein uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human SLC22A6 expressed in HEK293 cells in presence of para-aminohippuric acid/metforminMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of OAT1 (unknown origin)More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 3.90E+4nMAssay Description:TP_TRANSPORTER: inhibition of PHA uptake (PHA: 5uM) in hOAT1-expressing S2 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 4.31E+4nMAssay Description:Inhibition of OAT1 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 4.78E+4nMAssay Description:Inhibition of OAT1 (unknown origin)More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of OAT1 (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of Adefovir uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of OAT3 (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 6.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of 6-Carboxyfluorescein uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 8.30E+4nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in OAT-expressing OK cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 8.30E+4nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in OAT-expressing OK cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.27E+5nMAssay Description:TP_TRANSPORTER: inhibition of Urate uptake (Urate: 300 uM) in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair